The Effects Of Benzodiazepines And Its Effects On The Cell...

Xanax is a benzodiazepine that is most often used to treat anxiety. The effects of benzodiazepines mainly come from their ability to alter the movement of the inhibitory transmitter known as GABAa. GABA is triggered to release when it then can bind to the GABAa receptor. The binding of the two causes the ion channel to open and chloride ions are sent across the cell membrane. This causes the inhibitory factor by depolarizing the membrane (Griffin et al., 2013). Benzodiazepines are absorbed well through both per oral and parenteral administrations. However, absorption per orally is more rapid than any other route. Xanax in particular, is highly lipid soluble. Because it is highly lipid soluble, it means that it passes through the blood brain barrier more quickly. Xanax, otherwise known as alprazolam, reaches its peak in concentration in about one to two hours after administration (Griffin et al., 2013). The half-life, or the time it takes the drug to decrease by half, is about six to twenty-seven hours for adults (Griffin et al., 2013). There is a redistribution of benzodiazepines in body fat. This is a two phase process. During the first phase, there is a fast drop in the blood level as the drug is being redistributed throughout the body. During the second phase the blood level is more slow to drop than the first phase because the drug that is left in the blood is being metabolized and as that is happening it is being replaced by the drug t hat is being released from the bodyShow MoreRelatedDrugs and Society Essay925 Words   |  4 Pages1c. Describe the life cycle of a typical neurotransmitter. A cell membrane with the uptake of a particular precursor absorbs amino acids to create a neurotransmitter. The amino acids undergo synthesis with a reaction with enzymes to become a neurotransmitter. 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